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Lysine acetyltransferase inhibitors: structure-activity relationships and potential therapeutic implications

Francesco Fiorentino1, Antonello Mai2,3, Dante Rotili2

  • 1Department of Chemistry, University of Oxford, South Parks Road, Oxford OX1 3QZ, UK.

Future Medicinal Chemistry
|April 21, 2018
PubMed

Keywords:
KAT inhibitorscancerchemical probesco-crystal structureepigeneticsinhibitor kineticslysine acetyltransferasesstructure-based drug discovery

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