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Updated: Feb 11, 2026

Simultaneous Measurement of HDAC1 and HDAC6 Activity in HeLa Cells Using UHPLC-MS
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Published on: August 10, 2017

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Isoform-selective HDAC1/6/8 inhibitors with an imidazo-ketopiperazine cap containing stereochemical diversity

Bertrand Lecointre1, Remy Narozny2, Maria Teresa Borrello3

  • 1Normandie University, INSA Rouen, UNIROUEN, CNRS, COBRA (UMR 6014), 76000 Rouen, France.

Philosophical Transactions of the Royal Society of London. Series B, Biological Sciences
|April 25, 2018
PubMed

Keywords:
enzyme inhibitorsepigeneticshistone deacetylasespeptidomimeticszinc metalloenzymes

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