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Updated: Feb 11, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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2-Methylacrylamide as a bioisoster of thiourea group for 1,3-dibenzylthioureido TRPV1 receptor antagonists

Seol Rin Park1, Juhyun Kim1, Sun Young Lee1

  • 1College of Pharmacy, Sookmyung Women's University, Seoul 04310, South Korea.

Bioorganic & Medicinal Chemistry Letters
|May 1, 2018
PubMed

Keywords:
(45)Ca(2+)-Influx assay1,3-Dibenzylthioureas2-MethylacrylamideAntagonistBioisosterTRPV1

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