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Harnessing biosynthesis and quantitative NMR for late stage functionalization of lead molecules: Application to the

Michael A Brodney1, Raman Sharma2, John T Lazzaro2

  • 1Pfizer Worldwide Research and Development, 610 Main Street, Cambridge, MA 02139, United States.

Bioorganic & Medicinal Chemistry Letters
|May 3, 2018
PubMed

Keywords:
BiosynthesisLate-stage diversificationM1 positive allosteric modulator (PAM) programMedicinal chemistry design cycle

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