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Discovery of amino-1,4-oxazines as potent BACE-1 inhibitors

Siem Jakob Veenstra1, Heinrich Rueeger1, Markus Voegtle1

  • 1Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Pharma AG, CH-4057 Basel, Switzerland.

Bioorganic & Medicinal Chemistry Letters
|May 17, 2018
PubMed

Keywords:
Alzheimer’s diseaseAmino-1,4-oxazinesBACE-1P-gppK(a)

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