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A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9
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Small Molecule Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) Inhibitors: Hit to Lead Optimization of Systemic

Allyn T Londregan1, Liuqing Wei1, Jun Xiao1

  • 1Pfizer Medicinal Chemistry , Groton , Connecticut 06340 , United States.

Journal of Medicinal Chemistry
|June 8, 2018
PubMed

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