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Synthesis and biological evaluation of curcumin derivatives modified with α-amino boronic acid as proteasome

Wenjie Zhang1, Heyuan Bai1, Liqiang Han1

  • 1State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, PR China.

Bioorganic & Medicinal Chemistry Letters
|June 11, 2018
PubMed

Keywords:
Antitumor activityCurcumin derivativesProteasome inhibitorsSubunit selectivityα-Amino boronic acid

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