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Updated: Feb 9, 2026

Kinase Inhibitor Screening In Self-assembled Human Protein Microarrays
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Rational design of mitochondria-targeted pyruvate dehydrogenase kinase 1 inhibitors with improved selectivity and

Biao Xu1, Zhimei Yu1, Sichuan Xiang1

  • 1School of Pharmaceutical Sciences, Chongqing Key Laboratory of Natural Product Synthesis and Drug Research, Chongqing University, Chongqing, 401331, PR China.

European Journal of Medicinal Chemistry
|June 12, 2018
PubMed

Keywords:
Anti-cancer drugCancer metabolismCancer proliferationMitochondriaTriphenylphosphonium cation

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