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Updated: Feb 6, 2026

In vitro Reconstitution of the Active T. castaneum Telomerase
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In vitro Reconstitution of the Active T. castaneum Telomerase

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Ethenesulfonyl fluoride derivatives as telomerase inhibitors: structure-based design, SAR, and anticancer evaluation

Xing Chen1, Gao-Feng Zha2, Jie Quan Wang1

  • 1a School of Pharmacy, Anhui Province Key Laboratory of Major Autoimmune Diseases , Anhui Institute of Innovative Drugs, Anhui Medical University , Hefei , P. R. China.

Journal of Enzyme Inhibition and Medicinal Chemistry
|August 25, 2018
PubMed

Keywords:
Ethenesulfonyl fluorideinhibitorselective anticancer activitytelomerase

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