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Updated: Feb 4, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Synthesis of androgen receptor antagonists containing a pentafluorosulfanyl (SF5 ) moiety

Jiyu Jin1, Yan Zhou2, Dehua Yang2

  • 1Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, School of Chemistry and Molecular Engineering, East China Normal University, Shanghai, P. R. China.

Archiv Der Pharmazie
|October 16, 2018
PubMed

Keywords:
androgen receptorantagonistenzalutamidepentafluorosulfanyl

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