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Design, Synthesis and Characterization of Covalent KDM5 Inhibitors

Saleta Vazquez-Rodriguez1, Miranda Wright1,2, Catherine M Rogers1

  • 1Structural Genomics Consortium & Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford, OX3 7DQ and OX3 7FZ, UK.

Angewandte Chemie (International Ed. in English)
|November 16, 2018
PubMed

Keywords:
KDM5covalent inhibitorsepigeneticslysine demethylase

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