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Quantifying Agonist Activity at G Protein-coupled Receptors
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Synthesis and Evaluation of Novel Biased μ-Opioid-Receptor (μOR) Agonists

Mengjun Ma1, Jialin Sun2, Menghua Li3

  • 1State Key Laboratory of Toxicology and Medical Countermeasures, Beijing Institute of Pharmacology & Toxicology, 27 Tai-Ping Road, Beijing 100850, China. mengjunma@126.com.

Molecules (Basel, Switzerland)
|January 16, 2019
PubMed

Keywords:
Gi signaling pathwayPZM21structure–activity relationshipβ-arrestin-2 recruitmentμOR-biased agonist

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