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Novel PIKK inhibitor antibody-drug conjugates: Synthesis and anti-tumor activity

Dahui Zhou1, Jeffrey Casavant1, Edmund I Graziani1

  • 1Oncology Medicinal Chemistry, Pfizer Worldwide Research and Development, 445 Eastern Point Road, Groton, CT 06340, United States.

Bioorganic & Medicinal Chemistry Letters
|January 19, 2019
PubMed

Keywords:
ADCAntitumorHER2-expressing tumor cell linesNeolymphostinPIKK inhibitorTrastuzumab conjugates

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