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Method for Identifying Small Molecule Inhibitors of the Protein-protein Interaction Between HCN1 and TRIP8b
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Targeting S100 Calcium-Binding Proteins with Small Molecule Inhibitors

Paul T Wilder1,2, Kristen M Varney1,2, David J Weber3,4

  • 1Center for Biomolecular Therapeutics (CBT), Department of Biochemistry and Molecular Biology, University of Maryland School of Medicine, Baltimore, MD, USA.

Methods in Molecular Biology (Clifton, N.J.)
|February 3, 2019
PubMed

Keywords:
Calcium bindingCancerFluorescence polarization competition assayHigh-throughput screeningInhibitorsMelanomaProtein-protein interfaceS100 proteinS100A1S100BSmall molecule

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