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Updated: Jan 29, 2026

Synthesis of Protein Bioconjugates via Cysteine-maleimide Chemistry
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HFIP-promoted Michael reactions: direct para-selective C-H activation of anilines with maleimides

Bang Li1, Qi Mao, Jia Zhou

  • 1Department of Medicinal Chemistry, Jiangsu Key Laboratory of Neuropsychiatric Diseases and College of Pharmaceutical Sciences, Soochow University, 199 Ren-Ai Road, Suzhou, Jiangsu 215123, People's Republic of China. yena@suda.edu.cn.

Organic & Biomolecular Chemistry
|February 6, 2019
PubMed

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