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4,6-Substituted-1H-Indazoles as potent IDO1/TDO dual inhibitors

Lingling Yang1, Yang Chen1, Junlin He2

  • 1Department of Pharmaceutical Engineering, School of Food and Bioengineering, Xihua University, Chengdu 610039, China.

Bioorganic & Medicinal Chemistry
|February 19, 2019
PubMed

Keywords:
1H-IndazolesAntitumor activityCancer immunotherapyDual inhibitorIndoleamine 2,3-dioxygenase 1 (IDO1)Tryptophan 2,3-dioxygenase (TDO)

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