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Updated: Jan 27, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A patent update on cannabinoid receptor 1 antagonists (2015-2018)

George Amato1, Nayaab S Khan1, Rangan Maitra1

  • 1a Center for Drug Discovery , RTI International , RTP , NC , USA.

Expert Opinion on Therapeutic Patents
|March 21, 2019
PubMed
Abstract

Keywords:
CB1NASHantagonistcannabinoidendocannabinoidmetabolic syndromeobesityperipheral

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