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Updated: Jan 26, 2026

Characterization of G Protein-coupled Receptors by a Fluorescence-based Calcium Mobilization Assay
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Characterization of G Protein-coupled Receptors by a Fluorescence-based Calcium Mobilization Assay

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Time-Resolved FRET-Based Assays to Characterize G Protein-Coupled Receptor Hetero-oligomer Pharmacology

Joyce Heuninck1,2,3, Candide Hounsou1,2,3, Elodie Dupuis4

  • 1CNRS, UMR 5203, Institut de Génomique Fonctionnelle, Montpellier, France.

Methods in Molecular Biology (Clifton, N.J.)
|April 11, 2019
PubMed

Keywords:
Binding experimentFluorescent ligandG protein-coupled receptorHTRF®Homo- and hetero-oligomerizationLanthanideSelf-labeling enzymeTag-lite® screeningTerbiumTime-resolved FRET

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