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Updated: Jan 26, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Third-generation CDK inhibitors: A review on the synthesis and binding modes of Palbociclib, Ribociclib and

Melania Poratti1, Giovanni Marzaro1

  • 1Department of Pharmaceutical and Pharmacological Sciences, University of Padova, via Marzolo 5, I-35131, Padova, Italy.

European Journal of Medicinal Chemistry
|April 13, 2019
PubMed

Keywords:
AbemaciclibCDKsPalbociclibRibociclibSynthesisThird-generation inhibitors

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