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Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D3 Receptor (D3R) Ligand Promiscuity

Sean W Reilly1, Aladdin A Riad1, Chia-Ju Hsieh1

  • 1Department of Radiology , Perelman School of Medicine, University of Pennsylvania , Philadelphia , Pennsylvania 19104 , United States.

Journal of Medicinal Chemistry
|April 26, 2019
PubMed

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