Endothelin receptor antagonism during preeclampsia: a matter of timing?

Emilie Hitzerd1,2, Rugina I Neuman1,3, Katrina M Mirabito Colafella1,4,5

  • 1Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus Medical Center, Rotterdam, The Netherlands.

Insights

Endothelin receptor antagonists (ERAs) show promise for preeclampsia treatment but carry teratogenic risks. Human pregnancy cases suggest ERAs may be safe if used later in pregnancy, avoiding organogenesis.

Area of Science:

  • Obstetrics and Gynecology
  • Pharmacology
  • Developmental Toxicology

Background:

  • Preeclampsia (PE) is a serious pregnancy complication lacking effective treatments.
  • The endothelin system is implicated in PE pathophysiology, with experimental models showing benefit from endothelin receptor antagonists (ERAs).
  • Animal studies indicate ERAs pose significant teratogenic risks, particularly craniofacial malformations.

Purpose of the Study:

  • To review human pregnancy cases involving ERA exposure.
  • To critically assess the potential teratogenic effects of ERAs in pregnant women.
  • To evaluate the feasibility of ERA use for preeclampsia treatment.

Main Methods:

  • Systematic literature search yielding 18 articles.
  • Analysis of 39 reported cases of ERA exposure during human pregnancy.
  • Review of pregnancy outcomes, including termination, miscarriage, and congenital abnormalities.

Main Results:

  • Most exposures occurred in the first trimester; five cases involved later or throughout pregnancy.
  • Elective termination occurred in 31% of pregnancies, and 5% resulted in spontaneous miscarriage.
  • No fetal congenital abnormalities were reported in the remaining cases.

Conclusions:

  • ERA treatment for severe preeclampsia might be considered later in pregnancy after organogenesis to mitigate teratogenic risks.
  • Further third-trimester toxicology studies are essential to confirm drug safety.
  • Efficacy in alleviating maternal PE symptoms and impact on neonatal outcomes require further investigation.

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