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Updated: Jan 19, 2026

Detection of Orexin and Cannabinoid Receptor Co-localization in Diet-Induced Obese Zebrafish
02:31

Detection of Orexin and Cannabinoid Receptor Co-localization in Diet-Induced Obese Zebrafish

426

Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist

Robert B Laprairie1, Kiran Vemuri1, Edward L Stahl1

  • 1Departments of Molecular Medicine and Neuroscience, The Scripps Research Institute, Jupiter, Florida (R.B.L., E.L.S., J.-H.H., T.W.G., L.M.B.); Center for Drug Discovery and Departments of Chemistry and Chemical Biology and Pharmaceutical Sciences, Northeastern University, Boston, Massachusetts (K.V., A.K., A.M.); iHuman Institute, ShanghaiTech University, Shanghai, China (T.H., Y.W., Z.-J.L.); and Departments of Biological Sciences and Chemistry, Bridge Institute, Michelson Center for Convergent Bioscience, University of Southern California, Los Angeles, California (R.C.S.).

Molecular Pharmacology
|September 14, 2019
PubMed

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