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Progress on small-molecule proteolysis-targeting chimeras

Wenhai Huang1, Beibei Wang1, Zhimin Zhang1

  • 1Key Laboratory of Neuropsychiatric Drug Research of Zhejiang Province, Institute of Materia Medica, Zhejiang Academy of Medical Sciences, Hangzhou, Zhejiang Province 310013, PR China.

Future Medicinal Chemistry
|October 2, 2019
PubMed

Keywords:
E3 ligasesPROTACsdegraderinduced protein degradationsmall moleculesubiquitinproteasome system

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