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Quantifying Agonist Activity at G Protein-coupled Receptors
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The nature of efficacy at G protein-coupled receptors

Peishen Zhao1, Sebastian G B Furness1

  • 1Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria 3052, Australia.

Biochemical Pharmacology
|October 5, 2019
PubMed

Keywords:
Biased agonismCell signalingEfficacyG protein coupled receptors (GPCRs)Receptor structure-functionReceptor theorySignal transduction

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