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High-affinity sigma-1 (σ1) receptor ligands based on the σ1 antagonist PB212

Mauro Niso1, Philip D Mosier2, Roberta Marottoli1

  • 1Dipartimento di Farmacia-Scienze del Farmaco, Università degli Studi di Bari ALDO MORO, Via Orabona 4, I-70125 Bari, Italy.

Future Medicinal Chemistry
|October 22, 2019
PubMed

Keywords:
molecular modelingsigma ligandssigma-1 receptorsigma-1 receptors antagonistsstructure–affinity relationship

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