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Discovery of coumarin-based selective aldehyde dehydrogenase 1A1 inhibitors with glucose metabolism improving

Dailin Liang1, Yazhou Fan2, Zhou Yang1

  • 1Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Tongjiaxiang 24, Nanjing, 210009, China; Department of Medicinal Chemistry, China Pharmaceutical University, Tongjiaxiang 24, Nanjing, 210009, China.

European Journal of Medicinal Chemistry
|December 10, 2019
PubMed

Keywords:
ALDH1A1 inhibitorsCoumarin derivativesGlucose consumptionSynthesis

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