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Updated: Jan 1, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Heterotrimeric G Proteins as Therapeutic Targets in Drug Discovery

Jian Li1, Yang Ge1, Jun-Xiang Huang1

  • 1Guangdong Key Laboratory of Chiral Molecule and Drug Discovery, School of Pharmaceutical Sciences, Sun Yat-sen University, 510006 Guangzhou, Guangdong, P. R. China.

Journal of Medicinal Chemistry
|December 17, 2019
PubMed

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