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Design of Glycosyltransferase Inhibitors: Serine Analogues as Pyrophosphate Surrogates?

Shuai Wang1, Jose A Cuesta-Seijo2, Alexander Striebeck2

  • 1Institut de Chimie et Biochimie Moléculaires et Supramoléculaires, Laboratoire de Chimie Organique 2-Glycochimie, UMR 5246, CNRS and Université Claude Bernard Lyon 1, 43 Boulevard du 11 Novembre 1918, 69622, Villeurbanne, France.

Chempluschem
|January 25, 2020
PubMed

Keywords:
amino acidscarbohydratesclick chemistryglycosyltransferasesinhibition

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