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Multi-step parallel synthesis enabled optimization of benzofuran derivatives as pan-genotypic non-nucleoside

Dong Xiao1, Xing Dai1, Hong Liu1

  • 1Department of Medicinal Chemistry, Merck & Co., Inc., 2015 Galloping Hill Road, Kenilworth, NJ 07033, USA.

Bioorganic & Medicinal Chemistry Letters
|February 17, 2020
PubMed

Keywords:
Lead optimizationMulti-step parallel librariesNS5B NNI inhibitorsPan-genotypic potency

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