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Discovery and optimization of 2-aminopyridine derivatives as novel and selective JAK2 inhibitors

Xiangyu Ma1, Yanyan Diao1, Huan Ge1

  • 1Shanghai Key Laboratory of New Drug Design, School of Pharmacy, East China University of Science & Technology, Shanghai 200237, China.

Bioorganic & Medicinal Chemistry Letters
|March 4, 2020
PubMed

Keywords:
JAK2SARSBDDSelectivity

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