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Structure-Activity Relationship between Thiol Group-Trapping Ability of Morphinan Compounds with a Michael Acceptor

Noriki Kutsumura1,2, Yasuaki Koyama2, Tsuyoshi Saitoh1

  • 1International Institute for Integrative Sleep Medicine (WPI-IIIS), University of Tsukuba, 1-1-1 Tennodai, Tsukuba, Ibaraki 305-8575, Japan.

Molecules (Basel, Switzerland)
|March 6, 2020
PubMed

Keywords:
1H-NMR experimentsBNTXmechanism elucidationmorphinanδ opioid receptor antagonist

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