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Updated: Dec 26, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Development and Structural Evaluation of N-Alkylated trans-2-Phenylcyclopropylamine-Based LSD1 Inhibitors

Hideaki Niwa1,2,3, Shin Sato1,2,3, Noriko Handa1

  • 1RIKEN Systems and Structural Biology Center, Yokohama, 230-0045, Japan.

Chemmedchem
|March 14, 2020
PubMed

Keywords:
X-ray crystallographychromatinepigeneticshistone demethylaseinhibitorsnucleosomesprotein structures

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