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An Efficient Method for the Synthesis of Peptoids with Mixed Lysine-type/Arginine-type Monomers and Evaluation of Their Anti-leishmanial Activity
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Design, synthesis and antifungal activity of pterolactam-inspired amide Mannich bases

Anca-Elena Dascalu1, Alina Ghinet2, Emmanuelle Lipka3

  • 1Univ. Lille, Inserm, CHU Lille, Institut Pasteur de Lille, U1167 - RID-AGE - Facteurs de risque et déterminants moléculaires des maladies liées au vieillissement, F-59000 Lille, France; Laboratoire de Chimie Durable et Santé, Health & Environment Department, Team Sustainable Chemistry, Ecole des Hautes Etudes d'Ingénieur (HEI), Yncréa Hauts-de-France, 13 Rue de Toul, F-59046 Lille, France; UFR Pharmacie, Laboratoire de Chimie Analytique, BP 83, F-59006 Lille, France; 'Alexandru Ioan Cuza' University of Iasi, Faculty of Chemistry, Bd. Carol I nr. 11, 700506 Iasi, Romania.

Fitoterapia
|April 3, 2020
PubMed

Keywords:
Antifungal agentsBiological screeningN,N′-aminalN,O-acetalPterolactam

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