Discovery of CNS-Penetrant Apoptosis Signal-Regulating Kinase 1 (ASK1) Inhibitors

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Zhili Xin1, Martin K Himmelbauer1, J Howard Jones1

  • 1Medicinal Chemistry, Bioassays, Drug Metabolism and Pharmacokinetics, and Physical Biochemistry and Molecular Design, Biotherapeutic and Medicinal Sciences, Biogen, 225 Binney Street, Cambridge, Massachusetts 02142, United States.

ACS Medicinal Chemistry Letters
|April 16, 2020
PubMed

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