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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A cellular perspective of bias at G protein-coupled receptors

Thomas J Fernandez1, Monica De Maria1, Braden T Lobingier1

  • 1Department of Chemical Physiology and Biochemistry, Oregon Health and Sciences University, Portland, Oregon, USA.

Protein Science : a Publication of the Protein Society
|April 17, 2020
PubMed

Keywords:
GPCRagonist biasdesensitizationsignaling

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