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Structure-activity relationship study of DEL-22379: ERK dimerization inhibitors with increased safety

Yang Yang1, Yuanzheng Zhou1, Lei Tao1

  • 1Cancer Center, West China Hospital, Sichuan University and Collaborative Innovation Center for Biotherapy, Chengdu, Sichuan, China.

Molecular Diversity
|May 8, 2020
PubMed

Keywords:
Anti-cancer activityERK dimerization inhibitorIndolin-2-oneStructure–activity relationshipSynthesis

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