Related Experiment Video

Updated: Dec 20, 2025

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
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A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors

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Inhibitors in AKTion: ATP-competitive vs allosteric

Glorianne Lazaro1, Eleftherios Kostaras1, Igor Vivanco1

  • 1Division of Cancer Therapeutics, The Institute of Cancer Research, 15 Cotswold Rd., SM2 5NG London, U.K.

Biochemical Society Transactions
|May 27, 2020
PubMed
Abstract

Keywords:
AKTATP-competitiveallostericcancerinhibitors

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