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Novel µ opioid antagonists derived from the µ opioid agonists endomorphin and [Dmt1 ]DALDA (H-Dmt-D-Arg-Phe-Lys-NH2 )

Saijian Shi1, Jian Xu1, LingLing Feng1

  • 1School of Pharmacy, Nanjing Medical University, Nanjing, China.

Chemical Biology & Drug Design
|June 12, 2020
PubMed

Keywords:
[Dmt1]DALDAendomorphinmu opioid receptor antagonistsopioid activity profilesproline analogues

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