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Discovery of the potent non-steroidal glucocorticoid receptor modulator BAY 1003803 as clinical candidate

Markus Berger1, Ekkehard May2, Hartmut Rehwinkel1

  • 1Medicinal Chemistry Berlin, Research & Development, Pharmaceuticals, Bayer AG, D-13353 Berlin, Germany.

Bioorganic & Medicinal Chemistry Letters
|July 8, 2020
PubMed

Keywords:
Amino alcoholGlucocorticoidSEGRATransactivationTransrepression

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