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Discovery of carboxyl-containing biaryl ureas as potent RORγt inverse agonists

Nannan Sun1, Yafei Huang1, Mingcheng Yu1

  • 1Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.

European Journal of Medicinal Chemistry
|July 23, 2020
PubMed

Keywords:
Autoimmune diseasesBiaryl ureasInverse agonistsRORγtTh17 cells

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