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Discovery of nonpeptide 3,4-dihydroquinazoline-4-carboxamides as potent and selective sst2 agonists

Jian Zhao1, Shimiao Wang1, Sangdon Han1

  • 1Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, San Diego, CA 92121, United States.

Bioorganic & Medicinal Chemistry Letters
|August 3, 2020
PubMed

Keywords:
3,4-dihydroquinazoline-4-carboxamideAcromegalyNeuroendocrine tumorsSomatostatinSst2 agonist

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