Discovery of a benzimidazole series as the first highly potent and selective ACSL1 inhibitors

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Kyohei Hayashi1, Noriyasu Kondo1, Naoki Omori1

  • 1Pharmaceutical Research Division, Shionogi Pharmaceutical Research Center, 3-1-1 Futaba-cho, Toyonaka, Osaka 561-0825, Japan.

Bioorganic & Medicinal Chemistry Letters
|December 7, 2020
PubMed

Keywords:
ACSL1Acyl-CoABenzimidazoleFatty acidSAR

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