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Updated: Nov 26, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Allosteric binding sites at the receptor-lipid bilayer interface: novel targets for GPCR drug discovery

Ying Wang1, Zhengtian Yu2, Wen Xiao2

  • 1Department of Pathophysiology, Key Laboratory of Cell Differentiation and Apoptosis of Chinese Ministry of Education, Shanghai Jiao Tong University, School of Medicine, Shanghai, 200025, China.

Drug Discovery Today
|December 10, 2020
PubMed

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