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Structure-activity relationship studies of dipeptide-based hepsin inhibitors with Arg bioisosteres

Hongmok Kwon1, Hyunsoo Ha1, Hayoung Jeon1

  • 1College of Pharmacy, Korea University, 2511 Sejong-ro, Jochiwon-eup, Sejong 30019, Republic of Korea.

Bioorganic Chemistry
|December 18, 2020
PubMed

Keywords:
BioisostereDipeptideHepsinProstate cancerStructure-activity relationship

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