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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Tctex-1 augments G protein-coupled receptor-mediated Gs signaling by activating adenylyl cyclase

Masaki Saito1, Ayano Chiba2, Takeya Sato3

  • 1Department of Molecular Pharmacology, Tohoku University Graduate School of Medicine, Sendai, 980-8575, Japan; Department of Cellular Signaling, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, 980-8578, Japan.

Journal of Pharmacological Sciences
|December 28, 2020
PubMed

Keywords:
Adenylyl cyclaseCytoplasmic dynein light chain Tctex-1Parathyroid hormone receptor

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