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A novel [5.2.1]bicyclic amine is a potent analgesic without µ opioid activity

Tetsuji Noguchi1, Yuma Umezaki1, Rieko Takano1

  • 1Medicinal Chemistry Research Laboratories, R&D Division, Daiichi Sankyo Co., Ltd., 1-2-58 Hiromachi, Shinagawa-ku, Tokyo 140-8710, Japan.

Bioorganic & Medicinal Chemistry Letters
|January 17, 2021
PubMed

Keywords:
AnalgesicBicyclic amineNaloxoneNon-opioidTail flick test

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