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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Function-Oriented and Modular (+/-)-cis-Pseudoguaianolide Synthesis: Discovery of New Nrf2 Activators and NF-κB

Fabien Emmetiere1, Ranjala Ratnayake2, Henry A M Schares3

  • 1Department of Chemistry, University of Florida, PO Box 117200, Gainesville, FL, 32608, USA.

Chemistry (Weinheim an Der Bergstrasse, Germany)
|January 27, 2021
PubMed

Keywords:
NF-κB inhibitorsNrf2 activatorsenyne metathesismodular synthesispseudoguaianolides

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