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A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
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Structural Insights into JAK2 Inhibition by Ruxolitinib, Fedratinib, and Derivatives Thereof

Ryan R Davis1, Baoli Li1, Sang Y Yun2

  • 1Drug Discovery DepartmentMoffitt Cancer Center, Tampa, Florida 33612, United States.

Journal of Medicinal Chemistry
|February 11, 2021
PubMed

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