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Updated: Nov 17, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Development of Generic G Protein Peptidomimetics Able to Stabilize Active State Gs Protein-Coupled Receptors for

Morgane Mannes1, Charlotte Martin1, Sarah Triest2

  • 1Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, 1050, Brussels, Belgium.

Angewandte Chemie (International Ed. in English)
|February 17, 2021
PubMed

Keywords:
GPCRsallosteric modulatorsdrug discoveryfragment screeningpeptidomimetics

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