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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Nonsteroidal antiandrogens. Synthesis and structure-activity relationships of 3-substituted derivatives of

H Tucker1, J W Crook, G J Chesterson

  • 1Imperial Chemical Industries PLC, Pharmaceuticals Division, Macclesfield, Cheshire, Great Britain.

Journal of Medicinal Chemistry
|May 1, 1988
PubMed

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